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Kinetic Studies and Bioactivity of Potential Manzamine Prodrugs

The manzamines represent a class of marine natural products that show considerable promise in the control of malaria but generate GI distress in rodents when administered orally in high doses. In an effort to generate manzamine prodrugs with improved antimalarial activity and reduced GI toxicity, we...

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Detalles Bibliográficos
Publicado en:J Nat Prod
Main Authors: Shilabin, Abbas Gholipour, Kasanah, Noer, Tekwani, Babu L., Hamann, Mark T.
Formato: Artigo
Idioma:Inglês
Publicado: 2008
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4918903/
https://ncbi.nlm.nih.gov/pubmed/18598080
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/np800163u
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