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Structure–activity relationship studies of manzamine A: Amidation of positions 6 and 8 of the β-carboline moiety

Twenty manzamine amides were synthesized and evaluated for in vitro antimalarial and antimicrobial activities. The amides of manzamine A (1) showed significantly reduced cytotoxicity against Vero cells, although were less active than 1. The structure–activity analysis showed that linear, short alkyl...

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Détails bibliographiques
Publié dans:Bioorg Med Chem
Auteurs principaux: Wahba, Amir E., Peng, Jiangnan, Kudrimoti, Sucheta, Tekwani, Babu L., Hamann, Mark T.
Format: Artigo
Langue:Inglês
Publié: 2009
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4883699/
https://ncbi.nlm.nih.gov/pubmed/19833520
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2009.09.026
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