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Novel functionalized 5-(phenoxymethyl)-1,3-dioxane analogs exhibiting cytochrome P450 inhibition: a patent evaluation WO2015048311 (A1)

Cytochrome P450's (CYP's) constitute a diverse group of over 500 monooxygenase hemoproteins, catalyzing transformations that involve xenobiotic metabolism, steroidogenesis and other metabolic processes. Over-production of the steroid hormone cortisol is implicated in the progression of dis...

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Dettagli Bibliografici
Pubblicato in:Expert Opin Ther Pat
Autori principali: Schroeder, Richard L, Tram, Phan, Liu, Jiawang, Foroozesh, Maryam, Sridhar, Jayalakshmi
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4904732/
https://ncbi.nlm.nih.gov/pubmed/26514241
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1517/13543776.2016.1105217
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