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BET and BRAF inhibitors act synergistically against BRAF‐mutant melanoma

Despite major advances in the treatment of metastatic melanoma, treatment failure is still inevitable in most cases. Manipulation of key epigenetic regulators, including inhibition of Bromodomain and extra‐terminal domain (BET) family members impairs cell proliferation in vitro and tumor growth in v...

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Detalles Bibliográficos
Publicado en:Cancer Med
Main Authors: Paoluzzi, Luca, Hanniford, Douglas, Sokolova, Elena, Osman, Iman, Darvishian, Farbod, Wang, Jinhua, Bradner, James E., Hernando, Eva
Formato: Artigo
Idioma:Inglês
Publicado: John Wiley and Sons Inc. 2016
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC4867668/
https://ncbi.nlm.nih.gov/pubmed/27169980
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cam4.667
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