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Simultaneous quantitative determination of 5-aza-2′-deoxycytidine genomic incorporation and DNA demethylation by liquid chromatography tandem mass spectrometry as exposure-response measures of nucleoside analog DNA methyltransferase inhibitors

The epigenetic and anti-cancer activities of the nucleoside analog DNA methyltransferase (DNMT) inhibitors decitabine (5-aza-2′-deoxycytidine, DAC), azacitidine, and guadecitabine are thought to require cellular uptake, metabolism to 5-aza-2′-deoxycytidine triphosphate, and incorporation into DNA. T...

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Библиографические подробности
Опубликовано в: :J Chromatogr B Analyt Technol Biomed Life Sci
Главные авторы: Anders, Nicole M., Liu, Jianyong, Wanjiku, Teresia, Giovinazzo, Hugh, Zhou, Jianya, Vaghasia, Ajay, Nelson, William G., Yegnasubramanian, Srinivasan, Rudek, Michelle A.
Формат: Artigo
Язык:Inglês
Опубликовано: 2016
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4866886/
https://ncbi.nlm.nih.gov/pubmed/27082761
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.jchromb.2016.03.029
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