Cargando...

On the Selectivity of the Gα(q) Inhibitor UBO-QIC: A Comparison with the Gα(i) Inhibitor Pertussis Toxin

Gα(q) inhibitor UBO-QIC (FR900359) is becoming an important pharmacological tool, but its selectivity against other G proteins and their subunits, especially βγ, has not been well characterized. We examined UBO-QIC's effect on diverse signaling pathways mediated via various G protein-coupled re...

Descripción completa

Guardado en:
Detalles Bibliográficos
Publicado en:Biochem Pharmacol
Autores principales: Gao, Zhan-Guo, Jacobson, Kenneth A.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2016
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4839537/
https://ncbi.nlm.nih.gov/pubmed/26954502
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bcp.2016.03.003
Etiquetas: Agregar Etiqueta
Sin Etiquetas, Sea el primero en etiquetar este registro!