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Development of Small-molecule HIV Entry Inhibitors Specifically Targeting gp120 or gp41

Human immunodeficiency virus type 1 (HIV-1) envelope (Env) glycoprotein surface subunit gp120 and transmembrane subunit gp41 play important roles in HIV-1 entry, thus serving as key targets for the development of HIV-1 entry inhibitors. T20 peptide (enfuvirtide) is the first U.S. FDA-approved HIV en...

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Bibliografske podrobnosti
izdano v:Curr Top Med Chem
Main Authors: Lu, Lu, Yu, Fei, Cai, Lifeng, Debnath, Asim K., Jiang, Shibo
Format: Artigo
Jezik:Inglês
Izdano: 2016
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC4775441/
https://ncbi.nlm.nih.gov/pubmed/26324044
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