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Development of Small-molecule HIV Entry Inhibitors Specifically Targeting gp120 or gp41

Human immunodeficiency virus type 1 (HIV-1) envelope (Env) glycoprotein surface subunit gp120 and transmembrane subunit gp41 play important roles in HIV-1 entry, thus serving as key targets for the development of HIV-1 entry inhibitors. T20 peptide (enfuvirtide) is the first U.S. FDA-approved HIV en...

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Publicat a:Curr Top Med Chem
Autors principals: Lu, Lu, Yu, Fei, Cai, Lifeng, Debnath, Asim K., Jiang, Shibo
Format: Artigo
Idioma:Inglês
Publicat: 2016
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4775441/
https://ncbi.nlm.nih.gov/pubmed/26324044
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