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Comprehensive Analysis of Structure Activity Relationships of α-Ketoheterocycles as sn-1-Diacylglycerol Lipase α Inhibitors

Diacylglycerol lipase α (DAGLα) is responsible for the formation of the endocannabinoid 2-arachidonoylglycerol (2-AG) in the central nervous system. DAGLα inhibitors are required to study the physiological role of 2-AG. Previously, we identified the α-ketoheterocycles as potent and highly selective...

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Dettagli Bibliografici
Pubblicato in:J Med Chem
Autori principali: Janssen, Freek J., Baggelaar, Marc P., Hummel, Jessica J. A., Overkleeft, Herman S., Cravatt, Benjamin F., Boger, Dale L., van der Stelt, Mario
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4690813/
https://ncbi.nlm.nih.gov/pubmed/26584396
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.5b01627
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