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Design of a Fluorescent Ligand Targeting the S-adenosylmethioine Binding Site of the Histone Methyltransferase MLL1

The histone methyltransferase MLL1 has been linked to translocation-associated gene fusion in childhood leukemias and is an attractive drug target. High-throughput biochemical analysis of MLL1 methyltransferase activity requires the production of at least a trimeric complex of MLL1, RbBP5 and WDR5 t...

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Détails bibliographiques
Publié dans:Org Biomol Chem
Auteurs principaux: Luan, Yepeng, Blazer, Levi L., Hu, Hao, Hajian, Taraneh, Zhang, Jing, Wu, Hong, Houliston, Scott, Arrowsmith, Cheryl H., Vedadi, Masoud, Zheng, Yujun George
Format: Artigo
Langue:Inglês
Publié: 2016
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4689628/
https://ncbi.nlm.nih.gov/pubmed/26541578
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c5ob01794g
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