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Ligand tunnels in T. brucei and human CYP51: Insights for parasite-specific drug design

BACKGROUND: Cytochrome P450 sterol 14α-demethylase (CYP51) is an essential enzyme for sterol biosynthesis and a target for anti-parasitic drug design. However, the design of parasite-specific drugs that inhibit parasitic CYP51 without severe side effects remains challenging. The active site of CYP51...

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Bibliographische Detailangaben
Veröffentlicht in:Biochim Biophys Acta
Hauptverfasser: Yu, Xiaofeng, Nandekar, Prajwal, Mustafa, Ghulam, Cojocaru, Vlad, Lepesheva, Galina I., Wade, Rebecca C.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2015
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4689311/
https://ncbi.nlm.nih.gov/pubmed/26493722
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bbagen.2015.10.015
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