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Potent Triazole Bisphosphonate Inhibitor of Geranylgeranyl Diphosphate Synthase

[Image: see text] Studies of triazole bisphosphonates have resulted in identification of a potent inhibitor of geranylgeranyl diphosphate synthase (IC(50) = 45 nM) with very good selectivity for this enzyme over farnesyl diphosphate synthase (IC(50) = 28 μM). This compound also potently disrupts ger...

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Vydáno v:ACS Med Chem Lett
Hlavní autoři: Wills, Veronica S., Allen, Cheryl, Holstein, Sarah A., Wiemer, David F.
Médium: Artigo
Jazyk:Inglês
Vydáno: American Chemical Society 2015
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4677368/
https://ncbi.nlm.nih.gov/pubmed/26713103
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.5b00334
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