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Optimized Diazo Scaffold for Protein Esterification

[Image: see text] The O-alkylation of carboxylic acids with diazo compounds provides a means to esterify carboxylic acids in aqueous solution. A Hammett analysis of the reactivity of diazo compounds derived from phenylglycinamide revealed that the p-methylphenylglycinamide scaffold has an especially...

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Dettagli Bibliografici
Pubblicato in:Org Lett
Autori principali: Mix, Kalie A., Raines, Ronald T.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4670563/
https://ncbi.nlm.nih.gov/pubmed/25938936
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.orglett.5b00840
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