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In Vitro Metabolism of Montelukast by Cytochrome P450s and UDP-Glucuronosyltransferases

Montelukast has been recommended as a selective in vitro and in vivo probe of cytochrome P450 (P450) CYP2C8 activity, but its selectivity toward this enzyme remains unclear. We performed detailed characterization of montelukast metabolism in vitro using human liver microsomes (HLMs), expressed P450s...

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Détails bibliographiques
Publié dans:Drug Metab Dispos
Auteurs principaux: Cardoso, Josiane de Oliveira, Oliveira, Regina Vincenzi, Lu, Jessica Bo Li, Desta, Zeruesenay
Format: Artigo
Langue:Inglês
Publié: The American Society for Pharmacology and Experimental Therapeutics 2015
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC4658491/
https://ncbi.nlm.nih.gov/pubmed/26374173
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.115.065763
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