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The binding selectivity of vonoprazan (TAK-438) to the gastric H(+),K(+)−ATPase

BACKGROUND: The gastric H(+),K(+)-ATPase is the preferred target for acid suppression. Until recently, the only drugs that effectively inhibited this ATPase were the proton pump inhibitors (PPIs). PPIs are acid-activated prodrugs that require acid protection. Once acid activated, PPIs bind to cystei...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:Aliment Pharmacol Ther
Prif Awduron: Scott, David R., Munson, Keith B., Marcus, Elizabeth A., Lambrecht, Nils W. G., Sachs, George
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2015
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC4626316/
https://ncbi.nlm.nih.gov/pubmed/26423447
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/apt.13414
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