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Mesotrypsin Has Evolved Four Unique Residues to Cleave Trypsin Inhibitors as Substrates

Human mesotrypsin is highly homologous to other mammalian trypsins, and yet it is functionally unique in possessing resistance to inhibition by canonical serine protease inhibitors and in cleaving these inhibitors as preferred substrates. Arg-193 and Ser-39 have been identified as contributors to th...

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Pubblicato in:J Biol Chem
Autori principali: Alloy, Alexandre P., Kayode, Olumide, Wang, Ruiying, Hockla, Alexandra, Soares, Alexei S., Radisky, Evette S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Biochemistry and Molecular Biology 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4571878/
https://ncbi.nlm.nih.gov/pubmed/26175157
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M115.662429
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