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Structure-Function Basis of Attenuated Inverse Agonism of Angiotensin II Type 1 Receptor Blockers for Active-State Angiotensin II Type 1 Receptor

Ligand-independent signaling by the angiotensin II type 1 receptor (AT1R) can be activated in clinical settings by mechanical stretch and autoantibodies as well as receptor mutations. Transition of the AT1R to the activated state is known to lower inverse agonistic efficacy of clinically used AT1R b...

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Опубликовано в: :Mol Pharmacol
Главные авторы: Takezako, Takanobu, Unal, Hamiyet, Karnik, Sadashiva S., Node, Koichi
Формат: Artigo
Язык:Inglês
Опубликовано: The American Society for Pharmacology and Experimental Therapeutics 2015
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4551048/
https://ncbi.nlm.nih.gov/pubmed/26121982
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.115.099176
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