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A channelopathy mechanism revealed by direct calmodulin activation of TrpV4

Ca(2+)-calmodulin (CaM) regulates varieties of ion channels, including Transient Receptor Potential vanilloid subtype 4 (TrpV4). It has previously been proposed that internal Ca(2+) increases TrpV4 activity through Ca(2+)-CaM binding to a C-terminal Ca(2+)-CaM binding domain (CBD). We confirmed this...

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Detalhes bibliográficos
Publicado no:Proc Natl Acad Sci U S A
Main Authors: Loukin, Stephen H., Teng, Jinfeng, Kung, Ching
Formato: Artigo
Idioma:Inglês
Publicado em: National Academy of Sciences 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4522800/
https://ncbi.nlm.nih.gov/pubmed/26170305
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1510602112
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