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Targeting Individual GPCRs with Redesigned Nonvisual Arrestins

Numerous human diseases are caused by excessive signaling of mutant G protein-coupled receptors (GPCRs) or receptors that are overstimulated due to upstream signaling imbalances. The feasibility of functional compensation by arrestins with enhanced ability to quench receptor signaling was recently t...

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Detalhes bibliográficos
Publicado no:Handb Exp Pharmacol
Main Authors: Gimenez, Luis E., Vishnivetskiy, Sergey A., Gurevich, Vsevolod V.
Formato: Artigo
Idioma:Inglês
Publicado em: 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4516156/
https://ncbi.nlm.nih.gov/pubmed/24292829
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/978-3-642-41199-1_8
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