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Discovery, synthesis and structure-activity analysis of symmetrical 2,7-disubstituted fluorenones as urea transporter inhibitors

Kidney urea transporters are targets for development of small-molecule inhibitors with action as salt-sparing diuretics. A cell-based, functional high-throughput screen identified 2,7-bisacetamido fluorenone 3 as a novel inhibitor of urea transporters UT-A1 and UT-B. Here, we synthesized twenty-two...

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Publicado no:Medchemcomm
Main Authors: Lee, Sujin, Esteva-Font, Cristina, Phuan, Puay-Wah, Anderson, Marc O., Verkman, A.S
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4501499/
https://ncbi.nlm.nih.gov/pubmed/26191399
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C5MD00198F
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