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Using Substrate Specificity of Antiplasmin-Cleaving Enzyme for Fibroblast Activation Protein Inhibitor Design()
Circulating antiplasmin-cleaving enzyme (APCE), a prolyl-specific serine proteinase, is essentially identical to membrane-inserted fibroblast activation protein (FAP) that is transiently expressed during epithelial-derived cancer growth. Human precursive α(2)-antiplasmin (Met-α(2)AP), the only known...
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| Izdano u: | Biochemistry |
|---|---|
| Glavni autori: | , , , , |
| Format: | Artigo |
| Jezik: | Inglês |
| Izdano: |
2009
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| Teme: | |
| Online pristup: | https://ncbi.nlm.nih.gov/pmc/articles/PMC4470291/ https://ncbi.nlm.nih.gov/pubmed/19402713 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/bi900257m |
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