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Review of Tolvaptan’s Pharmacokinetic and Pharmacodynamic Properties and Drug Interactions

Tolvaptan is an arginine vasopressin (AVP) antagonist that acts to increase excretion of free water (aquaresis) in patients without introducing electrolyte abnormalities or worsening renal function. It works via blockade of vasopressin-2 receptors at the renal collecting duct. Since the approval of...

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Publicado en:J Clin Med
Autores principales: Bhatt, Purav R., McNeely, Elizabeth B., Lin, Tess E., Adams, Kirkwood F., Patterson, J. Herbert
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI 2014
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4470182/
https://ncbi.nlm.nih.gov/pubmed/26237603
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/jcm3041276
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