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Multidrug Resistance-Associated Protein 3 Plays an Important Role in Protection against Acute Toxicity of Diclofenac

Diclofenac (DCF) is a nonsteroidal anti-inflammatory drug commonly prescribed to reduce pain in acute and chronic inflammatory diseases. One of the main DCF metabolites is a reactive diclofenac acyl glucuronide (DCF-AG) that covalently binds to biologic targets and may contribute to adverse drug rea...

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Detalhes bibliográficos
Publicado no:Drug Metab Dispos
Main Authors: Scialis, Renato J., Csanaky, Iván L., Goedken, Michael J., Manautou, José E.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2015
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4468432/
https://ncbi.nlm.nih.gov/pubmed/25897176
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.114.061705
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