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Synthesis of carbon-14, carbon-13 and deuterium labeled forms of thioacetamide and thioacetamide S-oxide

Thioacetamide (TA) is a model hepatotoxin that undergoes metabolic activation via two successive S-oxidations. The ultimate toxic metabolite thioacetamide S,S-dioxide, or its tautomer acetimidoyl sulfinic acid CH(3)C(NH)SO(2)H, then acylates lysine side chains on cellular proteins leading to cellula...

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Bibliografski detalji
Izdano u:J Labelled Comp Radiopharm
Glavni autori: Sarma, Diganta, Hanzlik, Robert P.
Format: Artigo
Jezik:Inglês
Izdano: 2011
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4461141/
https://ncbi.nlm.nih.gov/pubmed/26069392
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/jlcr.1933
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