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Three-dimensional Structure of a Kunitz-type Inhibitor in Complex with an Elastase-like Enzyme

Elastase-like enzymes are involved in important diseases such as acute pancreatitis, chronic inflammatory lung diseases, and cancer. Structural insights into their interaction with specific inhibitors will contribute to the development of novel anti-elastase compounds that resist rapid oxidation and...

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Dettagli Bibliografici
Pubblicato in:J Biol Chem
Autori principali: García-Fernández, Rossana, Perbandt, Markus, Rehders, Dirk, Ziegelmüller, Patrick, Piganeau, Nicolas, Hahn, Ulrich, Betzel, Christian, Chávez, María de los Ángeles, Redecke, Lars
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Biochemistry and Molecular Biology 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4447985/
https://ncbi.nlm.nih.gov/pubmed/25878249
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.M115.647586
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