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Synthesis of carbocyclic nucleoside analogs with five-membered heterocyclic nucleobases

New carbocyclic nucleoside analogs with five-membered heterocyclic nucleobases were synthesized and evaluated as potential anti-HIV and anti-HCV agents. Among the synthesized carbocyclic nucleoside analogs, the pyrazole amide 15f exhibited modest selective anti-HIV-1 activity (EC(50) = 24 µM).

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Dettagli Bibliografici
Pubblicato in:Tetrahedron Lett
Autori principali: Cho, Jong hyun, Coats, Steven J., Schinazi, Raymond F.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2015
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4446795/
https://ncbi.nlm.nih.gov/pubmed/26028788
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tetlet.2015.01.051
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