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Dolutegravir Resistance Mutation R263K Cannot Coexist in Combination with Many Classical Integrase Inhibitor Resistance Substitutions

The new integrase strand transfer inhibitor (INSTI) dolutegravir (DTG) displays limited cross-resistance with older drugs of this class and selects for the R263K substitution in treatment-experienced patients. We performed tissue culture selections with DTG, using viruses resistant to older INSTIs a...

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Detaylı Bibliyografya
Yayımlandı:J Virol
Asıl Yazarlar: Anstett, Kaitlin, Mesplede, Thibault, Oliveira, Maureen, Cutillas, Vincent, Wainberg, Mark A.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: American Society for Microbiology 2015
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC4442391/
https://ncbi.nlm.nih.gov/pubmed/25653436
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/JVI.03485-14
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