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Design and Synthesis of Novel Arctigenin Analogues for the Amelioration of Metabolic Disorders

[Image: see text] Analogues of the natural product (−)-arctigenin, an activator of adenosine monophosphate activated protein kinase, were prepared in order to evaluate their effects on 2-deoxyglucose uptake in L6 myotubes and possible use in ameliorating metabolic disorders. Racemic arctigenin 2a wa...

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Publicado en:ACS Med Chem Lett
Autores principales: Duan, Shudong, Huang, Suling, Gong, Jian, Shen, Yu, Zeng, Limin, Feng, Ying, Ren, Wenming, Leng, Ying, Hu, Youhong
Formato: Artigo
Lenguaje:Inglês
Publicado: American Chemical Society 2015
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4416425/
https://ncbi.nlm.nih.gov/pubmed/25941553
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.5b00007
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