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Novel Peptidomimetics for Inhibition of HER2:HER3 Heterodimerization in HER2-Positive Breast Cancer

The current approach to treating HER2-overexpressed breast cancer is the use of monoclonal antibodies or a combination of antibodies with traditional chemotherapeutic agents or kinase inhibitors. Our approach is to target clinically validated HER2 domain IV with peptidomimetics and inhibit the prote...

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Dettagli Bibliografici
Pubblicato in:Chem Biol Drug Des
Autori principali: Kanthala, Shanthi, Banappagari, Sashikanth, Gokhale, Ameya, Liu, Yong-Yu, Xin, Gu, Zhao, Yunfeng, Jois, Seetharama
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4408264/
https://ncbi.nlm.nih.gov/pubmed/25346057
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cbdd.12453
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