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Mutations at Tyrosine 88, Lysine 92 and Tyrosine 470 of human dopamine transporter result in an attenuation of HIV-1 Tat-induced inhibition of dopamine transport

HIV-1 transactivator of transcription (Tat) protein disrupts the dopamine (DA) neurotransmission by inhibiting DA transporter (DAT) function, leading to increased neurocognitive impairment in HIV-1 infected individuals. Through integrated computational modeling and pharmacological studies, we have d...

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Detalhes bibliográficos
Publicado no:J Neuroimmune Pharmacol
Main Authors: Midde, Narasimha M., Yuan, Yaxia, Quizon, Pamela M., Sun, Wei-Lun, Huang, Xiaoqin, Zhan, Chang-Guo, Zhu, Jun
Formato: Artigo
Idioma:Inglês
Publicado em: 2015
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4388869/
https://ncbi.nlm.nih.gov/pubmed/25604666
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11481-015-9583-3
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