Wird geladen...

Design, Synthesis, and Protein Crystallography of Biaryltriazoles as Potent Tautomerase Inhibitors of Macrophage Migration Inhibitory Factor

[Image: see text] Optimization is reported for biaryltriazoles as inhibitors of the tautomerase activity of human macrophage migration inhibitory factor (MIF), a proinflammatory cytokine associated with numerous inflammatory diseases and cancer. A combined approach was taken featuring organic synthe...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Veröffentlicht in:J Am Chem Soc
Hauptverfasser: Dziedzic, Pawel, Cisneros, José A., Robertson, Michael J., Hare, Alissa A., Danford, Nadia E., Baxter, Richard H. G., Jorgensen, William L.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2015
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4386841/
https://ncbi.nlm.nih.gov/pubmed/25697265
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ja512112j
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!