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The nonpeptide WIN 64338 is a bradykinin B2 receptor antagonist.

We report the synthesis and in vitro biological activity of the nonpeptide bradykinin receptor antagonist WIN 64338, [[4-[[2-[[bis(cyclohexylamino)methylene]amino]-3-(2- naphthyl)-1-oxopropyl]amino]phenyl]methyl]tributylphosphonium chloride monohydrochloride. WIN 64338 inhibits [3H]-bradykinin bindi...

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Detalles Bibliográficos
Autores principales: Sawutz, D G, Salvino, J M, Dolle, R E, Casiano, F, Ward, S J, Houck, W T, Faunce, D M, Douty, B D, Baizman, E, Awad, M M
Formato: Artigo
Lenguaje:Inglês
Publicado: 1994
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC43854/
https://ncbi.nlm.nih.gov/pubmed/8197121
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