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Inhibiting EGFR Dimerization Using Triazolyl-Bridged Dimerization Arm Mimics

The epidermal growth factor receptor (EGFR) is overexpressed in multiple carcinomas and is the focus of a variety of targeted therapies. Here we report the design of peptide-based compounds that mimic the EGFR dimerization arm and inhibit allosteric activation of EGFR. These peptides are modified to...

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Dades bibliogràfiques
Publicat a:PLoS One
Autors principals: Hanold, Laura E., Oruganty, Krishnadev, Ton, Norman T., Beedle, Aaron M., Kannan, Natarajan, Kennedy, Eileen J.
Format: Artigo
Idioma:Inglês
Publicat: Public Library of Science 2015
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4366150/
https://ncbi.nlm.nih.gov/pubmed/25790232
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0118796
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