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Structural requirements for TLR7-selective signaling by 9-(4-piperidinylalkyl)-8-oxoadenine derivatives

We report the synthesis and biological evaluation of a new series of 8-oxoadenines substituted at the 9-position with a 4-piperidinylalkyl moiety. In vitro evaluation of the piperidinyl-substituted oxoadenines 3a–g in human TLR7- or TLR8-transfected HEK293 cells and in human PBMCs indicated that TLR...

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Bibliografiske detaljer
Udgivet i:Bioorg Med Chem Lett
Main Authors: Bazin, Hélène G., Li, Yufeng, Khalaf, Juhienah K., Mwakwari, Sandra, Livesay, Mark T., Evans, Jay T., Johnson, David A.
Format: Artigo
Sprog:Inglês
Udgivet: 2015
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4357173/
https://ncbi.nlm.nih.gov/pubmed/25698055
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2015.01.037
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