Загрузка...

Competitive Binding of a Benzimidazole to the Histone-Binding Pocket of the Pygo PHD Finger

[Image: see text] The Pygo-BCL9 complex is a chromatin reader, facilitating β-catenin-mediated oncogenesis, and is thus emerging as a potential therapeutic target for cancer. Its function relies on two ligand-binding surfaces of Pygo’s PHD finger that anchor the histone H3 tail methylated at lysine...

Полное описание

Сохранить в:
Библиографические подробности
Опубликовано в: :ACS Chem Biol
Главные авторы: Miller, Thomas C. R., Rutherford, Trevor J., Birchall, Kristian, Chugh, Jasveen, Fiedler, Marc, Bienz, Mariann
Формат: Artigo
Язык:Inglês
Опубликовано: American Chemical Society 2014
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC4330097/
https://ncbi.nlm.nih.gov/pubmed/25323450
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb500585s
Метки: Добавить метку
Нет меток, Требуется 1-ая метка записи!