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K(v)11.1 (hERG)-induced cardiotoxicity: a molecular insight from a binding kinetics study of prototypical K(v)11.1 (hERG) inhibitors

BACKGROUND AND PURPOSE: Drug-induced arrhythmia due to blockade of the K(v)11.1 channel (also known as the hERG K(+) channel) is a frequent side effect. Previous studies have primarily focused on equilibrium parameters, i.e. affinity or potency, of drug candidates at the channel. The aim of this stu...

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Publicat a:Br J Pharmacol
Autors principals: Yu, Z, IJzerman, A P, Heitman, L H
Format: Artigo
Idioma:Inglês
Publicat: BlackWell Publishing Ltd 2015
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC4301700/
https://ncbi.nlm.nih.gov/pubmed/25296617
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.12967
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