Načítá se...

K(v)11.1 (hERG)-induced cardiotoxicity: a molecular insight from a binding kinetics study of prototypical K(v)11.1 (hERG) inhibitors

BACKGROUND AND PURPOSE: Drug-induced arrhythmia due to blockade of the K(v)11.1 channel (also known as the hERG K(+) channel) is a frequent side effect. Previous studies have primarily focused on equilibrium parameters, i.e. affinity or potency, of drug candidates at the channel. The aim of this stu...

Celý popis

Uloženo v:
Podrobná bibliografie
Vydáno v:Br J Pharmacol
Hlavní autoři: Yu, Z, IJzerman, A P, Heitman, L H
Médium: Artigo
Jazyk:Inglês
Vydáno: BlackWell Publishing Ltd 2015
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4301700/
https://ncbi.nlm.nih.gov/pubmed/25296617
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.12967
Tagy: Přidat tag
Žádné tagy, Buďte první, kdo otaguje tento záznam!