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Issues in interpreting the in vivo activity of Aurora-A inhibitors

INTRODUCTION: Based on its role as a mitotic regulatory kinase, overexpressed and associated with aneuploidy in cancer, small molecule inhibitors have been developed for Aurora-A (AURKA) kinase. In preclinical and clinical assessments, these agents have shown efficacy in inducing stable disease or t...

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Detaylı Bibliyografya
Yayımlandı:Expert Opin Ther Targets
Asıl Yazarlar: Shagisultanova, Elena, Dunbrack, Roland L., Golemis, Erica A.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2014
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC4294965/
https://ncbi.nlm.nih.gov/pubmed/25384454
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1517/14728222.2014.981154
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