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μ-Opioid receptor activation and noradrenaline transport inhibition by tapentadol in rat single locus coeruleus neurons

BACKGROUND AND PURPOSE: Tapentadol is a novel analgesic that combines moderate μ-opioid receptor agonism and noradrenaline reuptake inhibition in a single molecule. Both mechanisms of action are involved in producing analgesia; however, the potency and efficacy of tapentadol in individual neurons ha...

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Bibliografiske detaljer
Udgivet i:Br J Pharmacol
Main Authors: Sadeghi, Mahsa, Tzschentke, Thomas M, Christie, MacDonald J
Format: Artigo
Sprog:Inglês
Udgivet: Blackwell Publishing Ltd 2015
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4292960/
https://ncbi.nlm.nih.gov/pubmed/24372103
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/bph.12566
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