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D-amino acid peptide residualizing agents bearing N-hydroxysuccinimido-and maleimido- functional groups and their application for trastuzumab radioiodination

INTRODUCTION: Proteins that undergo receptor-mediated endocytosis are subject to lysosomal degradation, requiring radioiodination methods that minimize loss of radioactivity from tumor cells after this process occurs. To accomplish this, we developed the residualizing radioiodination agent N(∊)-(3-[...

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Dettagli Bibliografici
Pubblicato in:Nucl Med Biol
Autori principali: Pruszynski, Marek, Koumarianou, Eftychia, Vaidyanathan, Ganesan, Chitneni, Satish, Zalutsky, Michael R.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4268387/
https://ncbi.nlm.nih.gov/pubmed/25240914
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.nucmedbio.2014.08.007
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