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Redundant kinase activation and resistance of EGFR-tyrosine kinase inhibitors

Epidermal growth factor receptor (EGFR) tyrosine kinase inhibitors (TKIs) have shown dramatic effects against that tumors harboring EGFR activating mutations in the EGFR intracytoplasmic tyrosine kinase domain and resulted in cell apoptosis. Unfortunately, a number of patients ultimately developed r...

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Detalles Bibliográficos
Publicado en:Am J Cancer Res
Autores principales: Luo, Min, Fu, Li-Wu
Formato: Artigo
Lenguaje:Inglês
Publicado: e-Century Publishing Corporation 2014
Materias:
Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC4266699/
https://ncbi.nlm.nih.gov/pubmed/25520855
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