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Fragment-Based Screening of the Bromodomain of ATAD2

[Image: see text] Cellular and genetic evidence suggest that inhibition of ATAD2 could be a useful strategy to treat several types of cancer. To discover small-molecule inhibitors of the bromodomain of ATAD2, we used a fragment-based approach. Fragment hits were identified using NMR spectroscopy, an...

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Veröffentlicht in:J Med Chem
Hauptverfasser: Harner, Mary J., Chauder, Brian A., Phan, Jason, Fesik, Stephen W.
Format: Artigo
Sprache:Inglês
Veröffentlicht: American Chemical Society 2014
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4255743/
https://ncbi.nlm.nih.gov/pubmed/25314628
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jm501035j
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