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Gene Variants in CYP2C19 Are Associated with Altered In Vivo Bupropion Pharmacokinetics but Not Bupropion-Assisted Smoking Cessation Outcomes

Bupropion is used clinically to treat depression and to promote smoking cessation. It is metabolized by CYP2B6 to its active metabolite hydroxybupropion, yet alterations in CYP2B6 activity have little impact on bupropion plasma levels. Furthermore, less than 10% of a bupropion dose is excreted as ur...

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Bibliografske podrobnosti
Main Authors: Zhu, Andy Z. X., Zhou, Qian, Cox, Lisa Sanderson, Ahluwalia, Jasjit S., Benowitz, Neal L., Tyndale, Rachel F.
Format: Artigo
Jezik:Inglês
Izdano: The American Society for Pharmacology and Experimental Therapeutics 2014
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC4201132/
https://ncbi.nlm.nih.gov/pubmed/25187485
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.114.060285
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