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Synthesis and Biological Evaluation of Largazole Analogues with Modified Surface Recognition Cap Groups

Several largazole analogues with modified surface recognition cap groups were synthesized and their HDAC inhibitory activities were determined. The C7-epimer 12 caused negligible inhibition of HDAC activity, failed to induce global histone 3 (H3) acetylation in the HCT116 colorectal cancer cell line...

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Autori principali: Bhansali, Pravin, Hanigan, Christin L., Perera, Lalith, Casero, Robert A., Viranga Tillekeratne, L. M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4188730/
https://ncbi.nlm.nih.gov/pubmed/25203782
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejmech.2014.09.009
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