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Biological Evaluation of New Largazole Analogues: Alteration of Macrocyclic Scaffold with Click Chemistry

[Image: see text] We report the design, synthesis, and biological evaluation of a new series of largazole analogues in which a 4-methylthiazoline moiety was replaced with a triazole and tetrazole ring, respectively. Compound 7 bearing a tetrazole ring was identified to show much better selectivity f...

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Bibliografische gegevens
Hoofdauteurs: Li, Xianlin, Tu, Zhenchao, Li, Hua, Liu, Chunping, Li, Zheng, Sun, Qiao, Yao, Yiwu, Liu, Jinsong, Jiang, Sheng
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: American Chemical Society 2012
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC4027506/
https://ncbi.nlm.nih.gov/pubmed/24900575
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/ml300371t
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