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Largazole Analogues Embodying Radical Changes in the Depsipeptide Ring: Development of a More Selective and Highly Potent Analogue

A number of analogues of the marine-derived histone deacetylase inhibitor largazole incorporating major structural changes in the depsipeptide ring were synthesized. Replacing the thiazole-thiazoline fragment of largazole with a bipyridine group gave analogue 7 with potent cell growth inhibitory act...

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Bibliografske podrobnosti
izdano v:J Med Chem
Main Authors: Almaliti, Jehad, Al-Hamashi, Ayad A., Negmeldin, Ahmed T., Hanigan, Christin L., Perera, Lalith, Pflum, Mary Kay H, Casero, Robert A., Viranga Tillekeratne, L. M.
Format: Artigo
Jezik:Inglês
Izdano: 2016
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC5574184/
https://ncbi.nlm.nih.gov/pubmed/27809521
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.6b01271
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