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Nigramide J is a novel potent inverse agonist of the human constitutive androstane receptor

The constitutive androstane receptor (CAR, NR1I3) is very important for drug development and for understanding pharmacokinetic drug–drug interactions. We screened by mammalian one hybrid assay among natural compounds to discover novel ligands of human constitutive androstane receptor (hCAR). hCAR tr...

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Detalhes bibliográficos
Main Authors: Kanno, Yuichiro, Tanuma, Nobuaki, Yatsu, Tomofumi, Li, Wei, Koike, Kazuo, Inouye, Yoshio
Formato: Artigo
Idioma:Inglês
Publicado em: Blackwell Publishing Ltd 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4186399/
https://ncbi.nlm.nih.gov/pubmed/25505573
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prp2.18
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