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Binding site multiplicity with fatty acid ligands: Implications for the regulation of PKR kinase autophosphorylation with palmitate

Saturated long chain-free fatty acids (FFAs), especially palmitate, have been implicated in apoptosis by inhibiting the activity of PKR (double-stranded RNA-dependent protein kinase). We recently found evidence that palmitate interacts directly with the kinase domain of PKR, subsequently inhibiting...

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Bibliografski detalji
Glavni autori: Fang, Liang, Cho, Hyun Ju, Chan, Christina, Feig, Michael
Format: Artigo
Jezik:Inglês
Izdano: 2014
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4177322/
https://ncbi.nlm.nih.gov/pubmed/24862841
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/prot.24607
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