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Synthesis of cell-permeable stapled BH3 peptide-based Mcl-1 inhibitors containing simple aryl and vinylaryl cross-linkers

We report the synthesis of a series of distance-matching aryl and vinylaryl cross-linkers for constructing stapled peptides containing cysteines at i,i+7 positions. Langevin dynamics simulation studies helped to classify these cross-linkers into two categories: the rigid cross-linkers with narrower...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Muppidi, Avinash, Doi, Kenichiro, Ramil, Carlo P., Wang, Hong-Gang, Lin, Qing
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2014
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4175436/
https://ncbi.nlm.nih.gov/pubmed/25267861
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tet.2014.05.104
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