A carregar...

Physicochemical Property-Driven Optimization of Diarylaniline Compounds as Potent HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors

Using physicochemical property-driven optimization, twelve new diarylaniline compounds (DAANs) (7a–h, 11a–b and 12a–b) were designed and synthesized. Among them, compounds 12a–b not only showed high potency (EC(50) 0.96–4.92 nM) against both wild-type and drug-resistant viral strains with the lowest...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Main Authors: Liu, Na, Qin, Bingjie, Sun, Lian-Qi, Yu, Fei, Lu, Lu, Jiang, Shibo, Lee, Kuo-Hsiung, Xie, Lan
Formato: Artigo
Idioma:Inglês
Publicado em: 2014
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC4137035/
https://ncbi.nlm.nih.gov/pubmed/25042339
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2014.07.011
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!